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Academic Journal

Design, synthesis and characterization of lead compounds as anti-inflammatory drugs targeting mPGES-1 via enzymelink screening.

  • Authors : Lu R; Department of Pharmacological & Pharmaceutical Sciences, Center for Experimental Therapeutics & Pharmacoinformatics, College of Pharmacy, University of Houston, Houston, TX 77204, USA.; Akasaka H

Subjects: Dinoprostone* ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/chemistry

  • Source: Future medicinal chemistry [Future Med Chem] 2023 May; Vol. 15 (9), pp. 757-767. Date of Electronic Publication: 2023 May 30.Publisher: Future Science Country of Publication: England NLM ID: 101511162 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Synthesis and Biological Evaluation of Gentiopicroside Derivatives as Novel Cyclooxygenase-2 Inhibitors with Anti-Inflammatory Activity.

  • Authors : Ren G; Gansu University of Chinese Medicine, Lanzhou, 730000, People's Republic of China.; Zhang Q

Subjects: Cyclooxygenase 2 Inhibitors*/Cyclooxygenase 2 Inhibitors*/Cyclooxygenase 2 Inhibitors*/chemistry ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/therapeutic use; Mice

  • Source: Drug design, development and therapy [Drug Des Devel Ther] 2023 Mar 23; Vol. 17, pp. 919-935. Date of Electronic Publication: 2023 Mar 23 (Print Publication: 2023).Publisher: Dove Press Limited Country of Publication: New Zealand NLM ID: 101475745 Publication Model: eCollection Cited Medium: Internet ISSN:

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Academic Journal

Nano-Phytopharmaceuticals in Inflammation.

  • Authors : Nair AS; Department of Pharmacognosy, KVM College of Pharmacy, Cherthala, Alappuzha (Dist.), Kerala, 688527, India.; Kopilakkal R

Subjects: Anti-Inflammatory Agents, Non-Steroidal* ; Synthetic Drugs*/Synthetic Drugs*/Synthetic Drugs*/therapeutic use; Humans

  • Source: Recent advances in inflammation & allergy drug discovery [Recent Adv Inflamm Allergy Drug Discov] 2023; Vol. 17 (1), pp. 31-38.Publisher: Bentham Science Publishers Country of Publication: Netherlands NLM ID: 101776469 Publication Model: Print Cited Medium: Internet ISSN:

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Academic Journal

Synthesis, In Vitro Anti-Inflammatory Activity, and HRMS Analysis of New Amphetamine Derivatives.

  • Authors : Manolov S; Department of Organic Chemistry, Faculty of Chemistry, University of Plovdiv, 4000 Plovdiv, Bulgaria.; Ivanov I

Subjects: Anti-Inflammatory Agents, Non-Steroidal*/Anti-Inflammatory Agents, Non-Steroidal*/Anti-Inflammatory Agents, Non-Steroidal*/pharmacology ; Anti-Inflammatory Agents, Non-Steroidal*/Anti-Inflammatory Agents, Non-Steroidal*/Anti-Inflammatory Agents, Non-Steroidal*/chemistry ; Ketoprofen*/Ketoprofen*/Ketoprofen*/chemistry

  • Source: Molecules (Basel, Switzerland) [Molecules] 2022 Dec 24; Vol. 28 (1). Date of Electronic Publication: 2022 Dec 24.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Constituents from the Polar Extract of Pisolithus arhizus and Their Anti-inflammatory Activity.

  • Authors : Parisi V; Dipartimento di Farmacia, Università degli Studi di Salerno, 84084 Fisciano (SA), Italy.; Nocera R

Subjects: Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/chemistry ; Triterpenes*/Triterpenes*/Triterpenes*/pharmacology Pisolithus arhizus

  • Source: Journal of natural products [J Nat Prod] 2024 Mar 22; Vol. 87 (3), pp. 520-529. Date of Electronic Publication: 2024 Feb 27.Publisher: American Society of Pharmacognosy Country of Publication: United States NLM ID: 7906882 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Benralizumab versus Mepolizumab for Eosinophilic Granulomatosis with Polyangiitis.

Subjects: Antibodies, Monoclonal, Humanized*/Antibodies, Monoclonal, Humanized*/Antibodies, Monoclonal, Humanized*/administration & dosage ; Antibodies, Monoclonal, Humanized*/Antibodies, Monoclonal, Humanized*/Antibodies, Monoclonal, Humanized*/adverse effects ; Antibodies, Monoclonal, Humanized*/Antibodies, Monoclonal, Humanized*/Antibodies, Monoclonal, Humanized*/pharmacology

  • Source: The New England journal of medicine [N Engl J Med] 2024 Mar 07; Vol. 390 (10), pp. 911-921. Date of Electronic Publication: 2024 Feb 23.Publisher: Massachusetts Medical Society Country of Publication: United States NLM ID: 0255562 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Celastrol regulates psoriatic inflammation and autophagy by targeting IL-17A.

  • Authors : Park A; Laboratory of PharmacoImmunology, Integrated Research Institute of Pharmaceutical Sciences and BK21 FOUR Team for Advanced Program for SmartPharma Leaders, College of Pharmacy, The Catholic University of Korea, 43 Jibong-ro, Bucheon-si, Gyeonggi-do 14662, Republic of Korea.; Heo TH

Subjects: Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/therapeutic use ; Interleukin-17*/Interleukin-17*/Interleukin-17*/antagonists & inhibitors

  • Source: Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie [Biomed Pharmacother] 2024 Mar; Vol. 172, pp. 116256. Date of Electronic Publication: 2024 Feb 16.Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 8213295 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Computational screening of potential anti-inflammatory leads from Jeevaneeya Rasayana plants targeting COX-2 and 5- LOX by molecular docking and dynamic simulation approaches.

  • Authors : Hemavathi KN; Center for Systems Biology and Molecular Medicine, Yenepoya Research Centre, Yenepoya (Deemed to be University), Mangalore, India.; Skariyachan S

Subjects: Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/chemistry ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/therapeutic use

  • Source: Computers in biology and medicine [Comput Biol Med] 2024 Mar; Vol. 171, pp. 108164. Date of Electronic Publication: 2024 Feb 15.Publisher: Elsevier Country of Publication: United States NLM ID: 1250250 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Design and synthesis of novel dithiazole carboxylic acid Derivatives: In vivo and in silico investigation of their Anti-Inflammatory and analgesic effects.

  • Authors : Yücel NT; Department of Pharmacology, Faculty of Pharmacy, Anadolu University, Eskişehir 26100, Turkey.; Asfour AAR

Subjects: Analgesics*/Analgesics*/Analgesics*/pharmacology ; Analgesics*/Analgesics*/Analgesics*/therapeutic use ; Analgesics*/Analgesics*/Analgesics*/chemistry

  • Source: Bioorganic chemistry [Bioorg Chem] 2024 Mar; Vol. 144, pp. 107120. Date of Electronic Publication: 2024 Jan 12.Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

The formyl peptide receptors FPR1 and FPR2 as targets for inflammatory disorders: recent advances in the development of small-molecule agonists.

  • Authors : Yi X; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, 3052, Australia.; Tran E

Subjects: Neutrophils* ; Receptors, Formyl Peptide*/Receptors, Formyl Peptide*/Receptors, Formyl Peptide*/agonists ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/chemistry

  • Source: European journal of medicinal chemistry [Eur J Med Chem] 2024 Feb 05; Vol. 265, pp. 115989. Date of Electronic Publication: 2023 Nov 27.Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet

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  • 10-20 of  295,160 results for ""ANTI-inflammatory agents""