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Academic Journal

Identification of a selective BRD4 PROTAC with potent antiproliferative effects in AR-positive prostate cancer based on a dual BET/PLK1 inhibitor.

  • Authors : Hu R; School of Life Science and Engineering, Southwest Jiaotong University, Chengdu, China.; Wang WL

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology ; Cell Cycle Proteins/Cell Cycle Proteins/Cell Cycle Proteins/*antagonists & inhibitors ; Prostatic Neoplasms/Prostatic Neoplasms/Prostatic Neoplasms/*drug therapy

  • Source: European journal of medicinal chemistry [Eur J Med Chem] 2022 Jan 05; Vol. 227, pp. 113922. Date of Electronic Publication: 2021 Oct 19.Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

BET inhibitor suppresses migration of human hepatocellular carcinoma by inhibiting SMARCA4.

  • Authors : Choi HI; Department of Bionanotechnology, Hanyang University, Seoul, 04673, Republic of Korea.; An GY

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology ; Carcinoma, Hepatocellular/Carcinoma, Hepatocellular/Carcinoma, Hepatocellular/*genetics ; DNA Helicases/DNA Helicases/DNA Helicases/*genetics

  • Source: Scientific reports [Sci Rep] 2021 Jun 03; Vol. 11 (1), pp. 11799. Date of Electronic Publication: 2021 Jun 03.Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

BET bromodomain-containing epigenetic reader proteins regulate vascular smooth muscle cell proliferation and neointima formation.

  • Authors : Dutzmann J; Mid-Germany Heart Center, Division of Cardiology, Angiology, and Intensive Medical Care, University Hospital Halle, Martin-Luther-University Halle-Wittenberg, Ernst-Grube-Straße 40, 06120 Halle, Germany.; Department of Cardiology and Angiology, Hannover Medical School, Carl-Neuberg-Str. 1, 30625 Hannover, Germany.

Subjects: Cell Proliferation*/Cell Proliferation*/Cell Proliferation*/drug effects ; Neointima*; Carotid Artery Injuries/Carotid Artery Injuries/Carotid Artery Injuries/*metabolism

  • Source: Cardiovascular research [Cardiovasc Res] 2021 Feb 22; Vol. 117 (3), pp. 850-862.Publisher: Oxford Journals Country of Publication: England NLM ID: 0077427 Publication Model: Print Cited Medium: Internet ISSN: 1755-3245

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Academic Journal

Double Mutant Cycles as a Tool to Address Folding, Binding, and Allostery.

  • Authors : Pagano L; Istituto Pasteur-Fondazione Cenci Bolognetti, Dipartimento di Scienze Biochimiche 'A. Rossi Fanelli' and Istituto di Biologia e Patologia Molecolari del CNR, Sapienza Università di Roma, 00185 Rome, Italy.; Toto A

Subjects: Allosteric Regulation* ; Mutation* ; Protein Folding*

  • Source: International journal of molecular sciences [Int J Mol Sci] 2021 Jan 15; Vol. 22 (2). Date of Electronic Publication: 2021 Jan 15.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

4-Acyl Pyrroles as Dual BET-BRD7/9 Bromodomain Inhibitors Address BETi Insensitive Human Cancer Cell Lines.

  • Authors : Hügle M; Institut für Pharmazeutische Wissenschaften, Albert-Ludwigs-Universität Freiburg, Hermann-Herder-Str. 8, D-79104 Freiburg, Germany.; Institut für Biochemie, Albert-Ludwigs-Universität Freiburg, Albertstr. 21, D-79104 Freiburg, Germany.

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*chemistry ; Chromosomal Proteins, Non-Histone/Chromosomal Proteins, Non-Histone/Chromosomal Proteins, Non-Histone/*antagonists & inhibitors ; Proteins/Proteins/Proteins/*antagonists & inhibitors

  • Source: Journal of medicinal chemistry [J Med Chem] 2020 Dec 24; Vol. 63 (24), pp. 15603-15620. Date of Electronic Publication: 2020 Dec 04.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Arabidopsis Transcription Factors SPL1 and SPL12 Confer Plant Thermotolerance at Reproductive Stage.

  • Authors : Chao LM; National Key Laboratory of Plant Molecular Genetics, CAS Center for Excellence in Molecular Plant Sciences, Shanghai Institute of Plant Physiology and Ecology, University of CAS, Chinese Academy of Sciences, Shanghai 200032, People's Republic of China.; Liu YQ

Subjects: Thermotolerance*; Arabidopsis/Arabidopsis/Arabidopsis/*physiology ; Arabidopsis Proteins/Arabidopsis Proteins/Arabidopsis Proteins/*physiology

  • Source: Molecular plant [Mol Plant] 2017 May 01; Vol. 10 (5), pp. 735-748. Date of Electronic Publication: 2017 Apr 08.Publisher: Cell Press Country of Publication: England NLM ID: 101465514 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Non-canonical transcriptional consequences of BET inhibition in cancer.

  • Authors : Letson C; Moffitt Cancer Center: 12902 USF Magnolia Drive, Tampa, FL 33612, United States. Electronic address: .; Padron E

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*therapeutic use ; Neoplasms/Neoplasms/Neoplasms/*drug therapy ; Proteins/Proteins/Proteins/*antagonists & inhibitors

  • Source: Pharmacological research [Pharmacol Res] 2019 Dec; Vol. 150, pp. 104508. Date of Electronic Publication: 2019 Nov 04.Publisher: Elsevier Country of Publication: Netherlands NLM ID: 8907422 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Cross-Species Genomics Reveals Oncogenic Dependencies in ZFTA/C11orf95 Fusion-Positive Supratentorial Ependymomas.

  • Authors : Zheng T; Hopp Children's Cancer Center Heidelberg (KiTZ), Heidelberg, Germany.; Division of Pediatric Neurooncology, German Cancer Research Center (DKFZ) and German Cancer Consortium (DKTK), Heidelberg, Germany.

Subjects: DNA-Binding Proteins/DNA-Binding Proteins/DNA-Binding Proteins/*genetics ; Ependymoma/Ependymoma/Ependymoma/*genetics ; Proteins/Proteins/Proteins/*genetics

  • Source: Cancer discovery [Cancer Discov] 2021 Sep; Vol. 11 (9), pp. 2230-2247. Date of Electronic Publication: 2021 Apr 20.Publisher: American Association for Cancer Research Country of Publication: United States NLM ID: 101561693 Publication Model: Print-Electronic Cited

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Academic Journal

Methylation‑driven genes PMPCAP1, SOWAHC and ZNF454 as potential prognostic biomarkers in lung squamous cell carcinoma.

  • Authors : Zhu Q; School of Medicine and Life Sciences, University of Jinan‑Shandong Academy of Medical Sciences, Jinan, Shandong 250022, P.R. China.; Wang J

Subjects: Carcinoma, Non-Small-Cell Lung/Carcinoma, Non-Small-Cell Lung/Carcinoma, Non-Small-Cell Lung/*diagnosis ; Carcinoma, Squamous Cell/Carcinoma, Squamous Cell/Carcinoma, Squamous Cell/*diagnosis ; DNA-Binding Proteins/DNA-Binding Proteins/DNA-Binding Proteins/*metabolism

  • Source: Molecular medicine reports [Mol Med Rep] 2020 Mar; Vol. 21 (3), pp. 1285-1295. Date of Electronic Publication: 2020 Jan 13.Publisher: D. A. Spandidos Country of Publication: Greece NLM ID: 101475259 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

An association study in the Taiwan Biobank elicits three novel candidates for cognitive aging in old adults: NCAM1, TTC12 and ZBTB20 .

  • Authors : Lin E; Department of Biostatistics, University of Washington, Seattle, WA 98195, USA.; Department of Electrical and Computer Engineering, University of Washington, Seattle, WA 98195, USA.

Subjects: Cognitive Aging* ; Polymorphism, Single Nucleotide*; CD56 Antigen/CD56 Antigen/CD56 Antigen/*genetics

  • Source: Aging [Aging (Albany NY)] 2021 Jul 20; Vol. 13 (14), pp. 18769-18788. Date of Electronic Publication: 2021 Jul 20.Publisher: Impact Journals, LLC Country of Publication: United States NLM ID: 101508617 Publication Model: Print-Electronic Cited Medium: Internet

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  • 1-10 of  51,573 results for ""TRANSCRIPTION factors""