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Academic Journal

A decade of USFDA-approved small molecules as anti-inflammatory agents: Recent trends and Commentaries on the "industrial" perspective.

  • Authors : Mehta V; Department of Cell Systems & Anatomy, University of Texas Health Science Center at San Antonio, Texas, 78229, USA.; Dwivedi AR

Subjects: Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/therapeutic use ; Signal Transduction*

  • Source: European journal of medicinal chemistry [Eur J Med Chem] 2024 Jan 05; Vol. 263, pp. 115942. Date of Electronic Publication: 2023 Nov 14.Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Synthesis and cytotoxic activity of ethyl ferulate derivatives as potent anti-inflammatory agents.

  • Authors : Fu DN; Medicinal Chemistry and Pharmacology Institute, Inner Mongolia Minzu University, Tongliao, Inner Mongolia, P.R. China.; Inner Mongolia Key Laboratory of Mongolian Medicine Pharmacology for Cardio-Cerebral Vascular System, Tongliao, Inner Mongolia, P.R. China.

Subjects: Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/therapeutic use ; Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/pharmacology

  • Source: Natural product research [Nat Prod Res] 2024 Jan-Feb; Vol. 38 (2), pp. 261-269. Date of Electronic Publication: 2022 Sep 02.Publisher: Taylor & Francis Health Sciences Country of Publication: England NLM ID: 101167924 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Design, synthesis, and biological investigation of oxadiazolyl, thiadiazolyl, and pyrimidinyl linked antipyrine derivatives as potential non-acidic anti-inflammatory agents.

  • Authors : Al-Sanea MM; Department of Pharmaceutical Chemistry, College of Pharmacy, Jouf University, Sakaka, Saudi Arabia.; Hamdi A

Subjects: Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Antipyrine*/Antipyrine*/Antipyrine*/pharmacology; Humans

  • Source: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2023 Dec; Vol. 38 (1), pp. 2162511.Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print Cited Medium: Internet ISSN: 1475-6374

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Academic Journal

Exploring new imines as anti-inflammatory COX and 5-LOX inhibitors with an improved pharmacokinetic profile.

  • Authors : Said MF; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Kasr El-Aini Street, Cairo, PO Box 11562, Egypt.; Moussa BA

Subjects: Tandem Mass Spectrometry* ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/therapeutic use

  • Source: Future medicinal chemistry [Future Med Chem] 2024 Feb; Vol. 16 (4), pp. 311-334. Date of Electronic Publication: 2024 Jan 31.Publisher: Future Science Country of Publication: England NLM ID: 101511162 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Investigations of new N 1 -substituted pyrazoles as anti-inflammatory and analgesic agents having COX inhibitory activity.

  • Authors : Said MF; Pharmaceutical Chemistry Department, Cairo University, Cairo, 11562, Egypt.; George RF

Subjects: Pyrazoles*/Pyrazoles*/Pyrazoles*/pharmacology ; Pyrazoles*/Pyrazoles*/Pyrazoles*/chemistry ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology

  • Source: Future medicinal chemistry [Future Med Chem] 2024 Feb; Vol. 16 (4), pp. 349-368. Date of Electronic Publication: 2024 Jan 30.Publisher: Future Science Country of Publication: England NLM ID: 101511162 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Methanesulfonamide derivatives as gastric safe anti-inflammatory agents: Design, synthesis, selective COX-2 inhibitory activity, histopathological and histochemical studies.

  • Authors : Abdelall EKA; Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.; Aboelnaga LS

Subjects: Cyclooxygenase 2 Inhibitors*/Cyclooxygenase 2 Inhibitors*/Cyclooxygenase 2 Inhibitors*/pharmacology ; Anti-Inflammatory Agents*; Cyclooxygenase 2

  • Source: Bioorganic chemistry [Bioorg Chem] 2023 Nov; Vol. 140, pp. 106787. Date of Electronic Publication: 2023 Aug 12.Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Fragment merging approach for the design of thiazole/thiazolidine clubbed pyrazoline derivatives as anti-inflammatory agents: Synthesis, biopharmacological evaluation and molecular modeling studies.

  • Authors : Elgohary MK; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Egyptian-Russian University, Badr City, Cairo 11829, Egypt.; Abd El Hadi SR

Subjects: Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Thiazoles*/Thiazoles*/Thiazoles*/pharmacology; Cyclooxygenase 2/Cyclooxygenase 2/Cyclooxygenase 2/metabolism

  • Source: Bioorganic chemistry [Bioorg Chem] 2023 Oct; Vol. 139, pp. 106724. Date of Electronic Publication: 2023 Jul 08.Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Discovery of Coixol Derivatives as Potent Anti-inflammatory Agents.

  • Authors : Cui E; College of Pharmacy, Anhui University of Chinese Medicine, Hefei 230012, China.; Qian S

Subjects: Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Signal Transduction*; Mice

  • Source: Journal of natural products [J Nat Prod] 2023 Aug 25; Vol. 86 (8), pp. 1950-1959. Date of Electronic Publication: 2023 Aug 10.Publisher: American Society of Pharmacognosy Country of Publication: United States NLM ID: 7906882 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Synthesis and anti-inflammatory activity of novel firocoxib analogues with balanced COX inhibition.

  • Authors : Xu J; Collaborative Innovation Center of Yangtze River Delta Region Green Pharmaceuticals, Zhejiang University of Technology, Hangzhou, China.; Tang K

Subjects: Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/chemistry ; Sulfones*/Sulfones*/Sulfones*/pharmacology

  • Source: Chemical biology & drug design [Chem Biol Drug Des] 2024 Jan; Vol. 103 (1), pp. e14437.Publisher: Wiley-Blackwell Country of Publication: England NLM ID: 101262549 Publication Model: Print Cited Medium: Internet ISSN: 1747-0285

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Academic Journal

Constituents from the Polar Extract of Pisolithus arhizus and Their Anti-inflammatory Activity.

  • Authors : Parisi V; Dipartimento di Farmacia, Università degli Studi di Salerno, 84084 Fisciano (SA), Italy.; Nocera R

Subjects: Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/chemistry ; Triterpenes*/Triterpenes*/Triterpenes*/pharmacology Pisolithus arhizus

  • Source: Journal of natural products [J Nat Prod] 2024 Mar 22; Vol. 87 (3), pp. 520-529. Date of Electronic Publication: 2024 Feb 27.Publisher: American Society of Pharmacognosy Country of Publication: United States NLM ID: 7906882 Publication Model: Print-Electronic Cited Medium:

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  • 1-10 of  422,903 results for ""Anti-Inflammatory Agents""