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Design, synthesis, and biological evaluation of a novel series of 1,2,4-oxadiazole inhibitors of SLACK potassium channels: Identification of in vitro tool VU0935685.

• Authors : Qunies AM; Department of Pharmaceutical Sciences, UNT System College of Pharmacy, University of North Texas Health Science Center, Fort Worth, TX 76107, USA; School of Biomedical Sciences, University of North Texas Health Science Center, Fort Worth, TX 76107, USA.

Subjects: Potassium Channels*/Potassium Channels*/Potassium Channels*/genetics ; Potassium Channels*/Potassium Channels*/Potassium Channels*/metabolism ; Thallium*/Thallium*/Thallium*/metabolism

• Source: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2023 Nov 15; Vol. 95, pp. 117487. Date of Electronic Publication: 2023 Sep 30.Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Discovery of a Small Molecule Activator of Slack (Kcnt1) Potassium Channels That Significantly Reduces Scratching in Mouse Models of Histamine-Independent and Chronic Itch.

• Authors : Balzulat A; Institute of Pharmacology and Clinical Pharmacy, Goethe University Frankfurt, Max-von-Laue-Str. 9, 60438, Frankfurt am Main, Germany.; Zhu WF

Subjects: Potassium Channels*/Potassium Channels*/Potassium Channels*/metabolism ; Potassium Channels*/Potassium Channels*/Potassium Channels*/therapeutic use ; Loxapine*/Loxapine*/Loxapine*/therapeutic use

• Source: Advanced science (Weinheim, Baden-Wurttemberg, Germany) [Adv Sci (Weinh)] 2024 Apr; Vol. 11 (15), pp. e2307237. Date of Electronic Publication: 2024 Feb 13.Publisher: WILEY-VCH Country of Publication: Germany NLM ID: 101664569 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2198-3844

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Modulation of potassium channels by transmembrane auxiliary subunits via voltage-sensing domains.

• Authors : Nakajo K; Division of Integrative Physiology, Department of Physiology, Jichi Medical University, Shimotsuke, Japan.; Kasuya G

Subjects: Potassium Channels* ; Ion Channels*; Binding Sites

• Source: Physiological reports [Physiol Rep] 2024 Mar; Vol. 12 (6), pp. e15980.Publisher: published by Wiley Periodicals, Inc. on behalf of the American Physiological Society and The Physiological Society Country of Publication: United States NLM

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Modelling and analysis of cAMP-induced mixed-mode oscillations in cortical neurons: Critical roles of HCN and M-type potassium channels.

• Authors : Martin M; Department of Information Engineering, University of Padova, Padova, Italy.; Pedersen MG

Subjects: Potassium Channels*/Potassium Channels*/Potassium Channels*/chemistry ; Nucleotides, Cyclic*/Nucleotides, Cyclic*/Nucleotides, Cyclic*/pharmacology; Neurons

• Source: PLoS computational biology [PLoS Comput Biol] 2024 Mar 22; Vol. 20 (3), pp. e1011559. Date of Electronic Publication: 2024 Mar 22 (Print Publication: 2024).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101238922 Publication Model: eCollection Cited Medium: Internet

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The potassium channels: Neurobiology and pharmacology of tinnitus.

• Authors : Lai H; Department of Otolaryngology, Sun Yat-sen Memorial Hospital, Sun Yat-sen University, Guangzhou, China.; Gao M

Subjects: Potassium Channels* ; Tinnitus*/Tinnitus*/Tinnitus*/drug therapy; Cricetinae

• Source: Journal of neuroscience research [J Neurosci Res] 2024 Jan; Vol. 102 (1), pp. e25281.Publisher: Wiley Interscience Country of Publication: United States NLM ID: 7600111 Publication Model: Print Cited Medium: Internet ISSN:

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CGP7930 - An allosteric modulator of GABA B Rs, GABA A Rs and inwardly-rectifying potassium channels.

• Authors : Hannan SB; Department of Neuroscience, Physiology and Pharmacology, University College London, Gower Street, London, WC1E 6BT, UK. Electronic address: .; Penzinger R

Subjects: Potassium Channels* ; Synaptic Transmission*; Rats

• Source: Neuropharmacology [Neuropharmacology] 2023 Nov 01; Vol. 238, pp. 109644. Date of Electronic Publication: 2023 Jul 06.Publisher: Pergamon Press Country of Publication: England NLM ID: 0236217 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Errata: Effect of Thimerosal on Arrhythmia Induced by Coronary Ligation: The Involvement of ATP-dependent Potassium Channels.

Subjects: Potassium Channels* ; Thimerosal*/Thimerosal*/Thimerosal*/pharmacology; Humans

• Source: International heart journal [Int Heart J] 2024; Vol. 65 (2), pp. 372.Publisher: International Heart Journal Association Country of Publication: Japan NLM ID: 101244240 Publication Model: Print Cited Medium: Internet

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Cycling matters: Sex hormone regulation of vascular potassium channels.

• Authors : Baldwin SN; Vascular Biology Group, Department of Biomedical Sciences, University of Copenhagen, Copenhagen, Denmark.; Jepps TA

Subjects: Progesterone* ; Potassium Channels*; Female

• Source: Channels (Austin, Tex.) [Channels (Austin)] 2023 Dec; Vol. 17 (1), pp. 2217637.Publisher: Taylor & Francis Country of Publication: United States NLM ID: 101321614 Publication Model: Print Cited Medium: Internet ISSN:

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Tongmai Yangxin pill alleviates myocardial no-reflow by activating GPER to regulate HIF-1α signaling and downstream potassium channels.

• Authors : Chen T; Key Laboratory of Hunan Province for Integrated Traditional Chinese and Western Medicine on Prevention and Treatment of Cardio-Cerebral Diseases, Hunan University of Chinese Medicine, Changsha, China.; Department of Clinical Pharmacology, Xiangya Hospital, Central South University, Changsha, People's Republic of China.

Subjects: NF-kappa B*/NF-kappa B*/NF-kappa B*/metabolism ; Potassium Channels*/Potassium Channels*/Potassium Channels*/metabolism; Animals

• Source: Pharmaceutical biology [Pharm Biol] 2023 Dec; Vol. 61 (1), pp. 499-513.Publisher: Taylor & Francis Country of Publication: England NLM ID: 9812552 Publication Model: Print Cited Medium: Internet ISSN: 1744-5116

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Kalium 3.0 is a comprehensive depository of natural, artificial, and labeled polypeptides acting on potassium channels.

• Authors : Krylov NA; Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.; Tabakmakher VM

Subjects: Potassium Channels*/Potassium Channels*/Potassium Channels*/genetics ; Databases, Pharmaceutical*; Ligands

• Source: Protein science : a publication of the Protein Society [Protein Sci] 2023 Nov; Vol. 32 (11), pp. e4776.Publisher: Cold Spring Harbor Laboratory Press Country of Publication: United States NLM ID: 9211750 Publication Model: Print Cited Medium: Internet

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