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Academic Journal

Binding of Gtf2i-β/δ transcription factors to the ARMS2 gene leads to increased circulating HTRA1 in AMD patients and in vitro.

  • Authors : Pan Y; Division of Molecular and Cellular Biology, National Institute of Sensory Organs, National Hospital Organization Tokyo Medical Center, Tokyo, Japan.; Iejima D

Subjects: High-Temperature Requirement A Serine Peptidase 1/High-Temperature Requirement A Serine Peptidase 1/High-Temperature Requirement A Serine Peptidase 1/*genetics ; Proteins/Proteins/Proteins/*genetics ; Transcription Factors, TFII/Transcription Factors, TFII/Transcription Factors, TFII/*genetics

  • Source: The Journal of biological chemistry [J Biol Chem] 2021 Jan-Jun; Vol. 296, pp. 100456. Date of Electronic Publication: 2021 Feb 24.Publisher: Elsevier Inc. on behalf of American Society for Biochemistry and Molecular Biology Country of Publication: United States NLM ID: 2985121R Publication

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Academic Journal

Identification of a selective BRD4 PROTAC with potent antiproliferative effects in AR-positive prostate cancer based on a dual BET/PLK1 inhibitor.

  • Authors : Hu R; School of Life Science and Engineering, Southwest Jiaotong University, Chengdu, China.; Wang WL

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology ; Cell Cycle Proteins/Cell Cycle Proteins/Cell Cycle Proteins/*antagonists & inhibitors ; Prostatic Neoplasms/Prostatic Neoplasms/Prostatic Neoplasms/*drug therapy

  • Source: European journal of medicinal chemistry [Eur J Med Chem] 2022 Jan 05; Vol. 227, pp. 113922. Date of Electronic Publication: 2021 Oct 19.Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

BET inhibitor suppresses migration of human hepatocellular carcinoma by inhibiting SMARCA4.

  • Authors : Choi HI; Department of Bionanotechnology, Hanyang University, Seoul, 04673, Republic of Korea.; An GY

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology ; Carcinoma, Hepatocellular/Carcinoma, Hepatocellular/Carcinoma, Hepatocellular/*genetics ; DNA Helicases/DNA Helicases/DNA Helicases/*genetics

  • Source: Scientific reports [Sci Rep] 2021 Jun 03; Vol. 11 (1), pp. 11799. Date of Electronic Publication: 2021 Jun 03.Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

BET bromodomain-containing epigenetic reader proteins regulate vascular smooth muscle cell proliferation and neointima formation.

  • Authors : Dutzmann J; Mid-Germany Heart Center, Division of Cardiology, Angiology, and Intensive Medical Care, University Hospital Halle, Martin-Luther-University Halle-Wittenberg, Ernst-Grube-Straße 40, 06120 Halle, Germany.; Department of Cardiology and Angiology, Hannover Medical School, Carl-Neuberg-Str. 1, 30625 Hannover, Germany.

Subjects: Cell Proliferation*/Cell Proliferation*/Cell Proliferation*/drug effects ; Neointima*; Carotid Artery Injuries/Carotid Artery Injuries/Carotid Artery Injuries/*metabolism

  • Source: Cardiovascular research [Cardiovasc Res] 2021 Feb 22; Vol. 117 (3), pp. 850-862.Publisher: Oxford Journals Country of Publication: England NLM ID: 0077427 Publication Model: Print Cited Medium: Internet ISSN: 1755-3245

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Academic Journal

Double Mutant Cycles as a Tool to Address Folding, Binding, and Allostery.

  • Authors : Pagano L; Istituto Pasteur-Fondazione Cenci Bolognetti, Dipartimento di Scienze Biochimiche 'A. Rossi Fanelli' and Istituto di Biologia e Patologia Molecolari del CNR, Sapienza Università di Roma, 00185 Rome, Italy.; Toto A

Subjects: Allosteric Regulation* ; Mutation* ; Protein Folding*

  • Source: International journal of molecular sciences [Int J Mol Sci] 2021 Jan 15; Vol. 22 (2). Date of Electronic Publication: 2021 Jan 15.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

4-Acyl Pyrroles as Dual BET-BRD7/9 Bromodomain Inhibitors Address BETi Insensitive Human Cancer Cell Lines.

  • Authors : Hügle M; Institut für Pharmazeutische Wissenschaften, Albert-Ludwigs-Universität Freiburg, Hermann-Herder-Str. 8, D-79104 Freiburg, Germany.; Institut für Biochemie, Albert-Ludwigs-Universität Freiburg, Albertstr. 21, D-79104 Freiburg, Germany.

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*chemistry ; Chromosomal Proteins, Non-Histone/Chromosomal Proteins, Non-Histone/Chromosomal Proteins, Non-Histone/*antagonists & inhibitors ; Proteins/Proteins/Proteins/*antagonists & inhibitors

  • Source: Journal of medicinal chemistry [J Med Chem] 2020 Dec 24; Vol. 63 (24), pp. 15603-15620. Date of Electronic Publication: 2020 Dec 04.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Profiling the regulatory interplay of BET bromodomains and Sirtuins in cancer cell lines.

Subjects: Azepines/Azepines/Azepines/*pharmacology ; Benzazepines/Benzazepines/Benzazepines/*pharmacology ; Benzodiazepines/Benzodiazepines/Benzodiazepines/*pharmacology

  • Source: Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie [Biomed Pharmacother] 2022 Mar; Vol. 147, pp. 112652. Date of Electronic Publication: 2022 Jan 19.Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 8213295 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

XP-524 is a dual-BET/EP300 inhibitor that represses oncogenic KRAS and potentiates immune checkpoint inhibition in pancreatic cancer.

  • Authors : Principe DR; Medical Scientist Training Program, University of Illinois College of Medicine, Chicago, IL 60612.; Department of Surgery, University of Illinois at Chicago, Chicago, IL 60612.

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology ; E1A-Associated p300 Protein/E1A-Associated p300 Protein/E1A-Associated p300 Protein/*antagonists & inhibitors ; Immune Checkpoint Inhibitors/Immune Checkpoint Inhibitors/Immune Checkpoint Inhibitors/*pharmacology

  • Source: Proceedings of the National Academy of Sciences of the United States of America [Proc Natl Acad Sci U S A] 2022 Jan 25; Vol. 119 (4).Publisher: National Academy of Sciences Country of Publication: United States NLM ID: 7505876 Publication Model: Print Cited Medium: Internet ISSN:

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Academic Journal

A paradigm shift in structural biology.

  • Authors : Subramaniam S; University of British Columbia, Vancouver, BC, Canada. .; Gandeeva Therapeutics Inc, Vancouver, BC, Canada. .

Subjects: Algorithms* ; Databases, Protein*/Databases, Protein*/Databases, Protein*/statistics & numerical data ; Models, Molecular*

  • Source: Nature methods [Nat Methods] 2022 Jan; Vol. 19 (1), pp. 20-23.Publisher: Nature Pub. Group Country of Publication: United States NLM ID: 101215604 Publication Model: Print Cited Medium: Internet ISSN:

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Academic Journal

Recent Developments in PROTAC-Mediated Protein Degradation: From Bench to Clinic.

  • Authors : Hu Z; Department of Molecular, Cellular and Developmental Biology, Yale University, 260 Whitney Avenue, New Haven, CT 06511, USA.; Crews CM

Subjects: Proteins/Proteins/Proteins/*metabolism; HeLa Cells ; Humans

  • Source: Chembiochem : a European journal of chemical biology [Chembiochem] 2022 Jan 19; Vol. 23 (2), pp. e202100270. Date of Electronic Publication: 2021 Sep 23.Publisher: Wiley-VCH Verlag Country of Publication: Germany NLM ID: 100937360 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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  • 1-10 of  19,105 results for ""TRANSCRIPTION factors""