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Academic Journal

Evo312: An Evodiamine Analog and Novel PKCβI Inhibitor with Potent Antitumor Activity in Gemcitabine-Resistant Pancreatic Cancer.

  • Authors : Bae ES; Natural Products Research Institute, College of Pharmacy, Seoul National University, Seoul 08826, Republic of Korea.; Hong J

Subjects: Pancreatic Neoplasms*/Pancreatic Neoplasms*/Pancreatic Neoplasms*/drug therapy ; Pancreatic Neoplasms*/Pancreatic Neoplasms*/Pancreatic Neoplasms*/pathology ; Gemcitabine*

  • Source: Journal of medicinal chemistry [J Med Chem] 2024 Sep 12; Vol. 67 (17), pp. 14885-14911. Date of Electronic Publication: 2024 Aug 16.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic

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Academic Journal

Extraction, Purification, Structural Characterization, and Antitumor Effects of Water-Soluble Intracellular Polysaccharide (IPSW-1) from Phellinus igniarius Mycelia.

  • Authors : Boateng ID; School of Food & Biological Engineering, Jiangsu University, Zhenjiang 212013, China.; Certified Group, 199 W Rhapsody Dr, San Antonio, Texas 78216, United States.

Subjects: Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/pharmacology ; Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/chemistry ; Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/isolation & purification

  • Source: Journal of agricultural and food chemistry [J Agric Food Chem] 2024 Sep 11; Vol. 72 (36), pp. 19721-19732. Date of Electronic Publication: 2024 Aug 29.Publisher: American Chemical Society Country of Publication: United States NLM ID: 0374755 Publication Model: Print-Electronic

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Academic Journal

New CDDO Arylboronate Ester Derivatives with High Selectivity and Low Toxicity.

  • Authors : Li N; State Key Laboratory of Natural Medicines, Department of Natural Medicinal Chemistry, School of Traditional Chinese Pharmacy, China Pharmaceutical University, 639 Longmian Avenue, Nanjing 211198, China.; Sate Key Laboratory for Chemistry and Molecular Engineering of Medicinal Resources, Guangxi Normal University, 15 Yucai Road, Guilin 541004, China.

Subjects: Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/pharmacology ; Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/chemistry ; Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/chemical synthesis

  • Source: Journal of medicinal chemistry [J Med Chem] 2024 Aug 22; Vol. 67 (16), pp. 14329-14344. Date of Electronic Publication: 2024 Aug 02.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic

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Academic Journal

Eurochevalierines A - I, Sesquiterpene Alkaloid Hybrids with Anti-Triple Negative Breast Cancer Activity from Penicillium sp. HZ-5.

  • Authors : Zhang Y; Hubei Key Laboratory of Natural Medicinal Chemistry and Resource Evaluation, Tongji Medical College, Huazhong University of Science and Technology, Wuhan 430030, China.; Li Q

Subjects: Penicillium*/Penicillium*/Penicillium*/chemistry ; Triple Negative Breast Neoplasms*/Triple Negative Breast Neoplasms*/Triple Negative Breast Neoplasms*/drug therapy ; Sesquiterpenes*/Sesquiterpenes*/Sesquiterpenes*/pharmacology

  • Source: Journal of agricultural and food chemistry [J Agric Food Chem] 2024 Jul 31; Vol. 72 (30), pp. 16801-16811. Date of Electronic Publication: 2024 Jul 17.Publisher: American Chemical Society Country of Publication: United States NLM ID: 0374755 Publication Model: Print-Electronic

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Academic Journal

Exploring the Potential of Cyclic Peptidyl Antitumor Agents Derived from Natural Macrocyclic Peptide Phakellistatin 13 .

  • Authors : Li T; Key Laboratory for Photonic and Electronic Bandgap Materials, Ministry of Education, College of Chemistry & Chemical Engineering, Harbin Normal University, Harbin 150025, China.; Jiang S

Subjects: Peptides, Cyclic*/Peptides, Cyclic*/Peptides, Cyclic*/chemistry ; Peptides, Cyclic*/Peptides, Cyclic*/Peptides, Cyclic*/pharmacology ; Peptides, Cyclic*/Peptides, Cyclic*/Peptides, Cyclic*/chemical synthesis

  • Source: Journal of medicinal chemistry [J Med Chem] 2024 Jul 25; Vol. 67 (14), pp. 11789-11813. Date of Electronic Publication: 2024 Jul 11.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic

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Academic Journal

Exploring the Health Benefits of Boletus aereus Polysaccharides: Extraction, Structural Characterization, and Antiproliferative Properties against Non-Hodgkin's Lymphomas (NHLs).

  • Authors : Wang H; Department of Urology, Institute of Urology (Laboratory of Reconstructive Urology), West China Hospital, Sichuan University, Chengdu 610041, China.; Faculty of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming 650500, China.

Subjects: Cell Proliferation*/Cell Proliferation*/Cell Proliferation*/drug effects ; Apoptosis*/Apoptosis*/Apoptosis*/drug effects ; Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/pharmacology

  • Source: Journal of agricultural and food chemistry [J Agric Food Chem] 2024 Jul 24; Vol. 72 (29), pp. 16334-16346. Date of Electronic Publication: 2024 Jul 12.Publisher: American Chemical Society Country of Publication: United States NLM ID: 0374755 Publication Model: Print-Electronic

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Academic Journal

β-Sitosterol Inhibits Tumor Growth and Amplifies Rituximab Sensitivity through Acid Sphingomyelinase/Ceramide Signaling in Diffuse Large B-Cell Lymphoma.

  • Authors : He G; Department of Oncology, Tianjin Union Medical Center of Nankai University, Tianjin 300121, China.; Department of Geriatrics, Binhai New Area Hospital of Traditional Chinese Medicine, Tianjin 300121, China.

Subjects: Lymphoma, Large B-Cell, Diffuse*/Lymphoma, Large B-Cell, Diffuse*/Lymphoma, Large B-Cell, Diffuse*/drug therapy ; Lymphoma, Large B-Cell, Diffuse*/Lymphoma, Large B-Cell, Diffuse*/Lymphoma, Large B-Cell, Diffuse*/metabolism ; Sphingomyelin Phosphodiesterase*/Sphingomyelin Phosphodiesterase*/Sphingomyelin Phosphodiesterase*/metabolism

  • Source: Journal of agricultural and food chemistry [J Agric Food Chem] 2024 Jul 24; Vol. 72 (29), pp. 16177-16190. Date of Electronic Publication: 2024 Jul 11.Publisher: American Chemical Society Country of Publication: United States NLM ID: 0374755 Publication Model: Print-Electronic

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Academic Journal

Development of Degraders of Cyclin-Dependent Kinases 4 and 6 Based on Rational Drug Design.

  • Authors : He H; Innovation Center for AI and Drug Discovery (ICAIDD), East China Normal University, Shanghai 200062, China.; Shanghai Key Laboratory of New Drug Design, School of Pharmacy, East China University of Science and Technology, Shanghai 200237, China.

Subjects: Drug Design* ; Cyclin-Dependent Kinase 4*/Cyclin-Dependent Kinase 4*/Cyclin-Dependent Kinase 4*/antagonists & inhibitors ; Cyclin-Dependent Kinase 4*/Cyclin-Dependent Kinase 4*/Cyclin-Dependent Kinase 4*/metabolism

  • Source: Journal of medicinal chemistry [J Med Chem] 2024 Jul 11; Vol. 67 (13), pp. 11354-11364. Date of Electronic Publication: 2024 Jun 29.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic

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Academic Journal

Carrier-Free Self-Assembled Nanomedicines for Promoting Apoptosis and Inhibiting Proliferation in Hepatocellular Carcinoma.

  • Authors : Jia W; Medical School, Southeast University, Nanjing 210009, China.; Yang M

Subjects: Apoptosis*/Apoptosis*/Apoptosis*/drug effects ; Carcinoma, Hepatocellular*/Carcinoma, Hepatocellular*/Carcinoma, Hepatocellular*/drug therapy ; Carcinoma, Hepatocellular*/Carcinoma, Hepatocellular*/Carcinoma, Hepatocellular*/pathology

  • Source: ACS biomaterials science & engineering [ACS Biomater Sci Eng] 2024 Jul 08; Vol. 10 (7), pp. 4347-4358. Date of Electronic Publication: 2024 Jun 06.Publisher: American Chemical Society Country of Publication: United States NLM ID: 101654670 Publication Model: Print-Electronic

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Academic Journal

Circ_002033 Regulates Proliferation, Apoptosis, and Oxidative Damage of Bovine Mammary Epithelial Cells via the miR-199a-5p-MAP3K11 Axis in Heat Stress.

  • Authors : Zeng H; College of Animal Science and Technology, Nanjing Agricultural University, Nanjing 210095, China.; Li S

Subjects: Epithelial Cells*/Epithelial Cells*/Epithelial Cells*/metabolism ; MicroRNAs*/MicroRNAs*/MicroRNAs*/genetics ; MicroRNAs*/MicroRNAs*/MicroRNAs*/metabolism

  • Source: Journal of agricultural and food chemistry [J Agric Food Chem] 2024 Jun 26; Vol. 72 (25), pp. 14386-14401. Date of Electronic Publication: 2024 Jun 13.Publisher: American Chemical Society Country of Publication: United States NLM ID: 0374755 Publication Model: Print-Electronic

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