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Academic Journal

Design, synthesis and biological evaluation of thiazolyl-halogenated pyrroles or pyrazoles as novel antibacterial and antibiofilm agents.

  • Authors : Zhong Y; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai, 201203, China; Department of Chemistry, Shanghai University, Shanghai 200444, China.

Subjects: Pyrazoles*/Pyrazoles*/Pyrazoles*/pharmacology ; Anti-Bacterial Agents*/Anti-Bacterial Agents*/Anti-Bacterial Agents*/pharmacology; Animals

  • Source: European journal of medicinal chemistry [Eur J Med Chem] 2024 Mar 15; Vol. 268, pp. 116221. Date of Electronic Publication: 2024 Feb 15.Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Investigations of new N 1 -substituted pyrazoles as anti-inflammatory and analgesic agents having COX inhibitory activity.

  • Authors : Said MF; Pharmaceutical Chemistry Department, Cairo University, Cairo, 11562, Egypt.; George RF

Subjects: Pyrazoles*/Pyrazoles*/Pyrazoles*/pharmacology ; Pyrazoles*/Pyrazoles*/Pyrazoles*/chemistry ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology

  • Source: Future medicinal chemistry [Future Med Chem] 2024 Feb; Vol. 16 (4), pp. 349-368. Date of Electronic Publication: 2024 Jan 30.Publisher: Future Science Country of Publication: England NLM ID: 101511162 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

"Antibacterial properties of nine indium(III) complexes of substituted pyrazoles/pyrazolate and the structural and solution characterization of the mer- and trans‑indium(III) complexes of 4-Me-pzH".

  • Authors : Herrera S; Department of Chemistry & Biochemistry and the Biomolecular Sciences Institute, Florida International University, Miami, FL 33199, USA.; Yoshinaga M

Subjects: Pyrazoles*/Pyrazoles*/Pyrazoles*/pharmacology ; Pyrazoles*/Pyrazoles*/Pyrazoles*/chemistry ; Indium*

  • Source: Journal of inorganic biochemistry [J Inorg Biochem] 2024 Jan; Vol. 250, pp. 112402. Date of Electronic Publication: 2023 Oct 14.Publisher: Elsevier Country of Publication: United States NLM ID: 7905788 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Design and synthesis of some novel hybrid molecules based on 4-thiazolidinone bearing pyridine-pyrazole scaffolds: molecular docking and molecular dynamics simulations of its major constituent onto DNA gyrase inhibition.

  • Authors : Desai NC; Division of Medicinal Chemistry, Department of Chemistry, Maharaja Krishnakumarsinhji Bhavnagar University, Mahatma Gandhi Campus, Bhavnagar, 364 002, India. .; Jadeja DJ

Subjects: Molecular Docking Simulation* ; Drug Design* ; Molecular Dynamics Simulation*

  • Source: Molecular diversity [Mol Divers] 2024 Apr; Vol. 28 (2), pp. 693-709. Date of Electronic Publication: 2023 Feb 08.Publisher: ESCOM Science Publishers Country of Publication: Netherlands NLM ID: 9516534 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Exploring Subsite Selectivity within Plasmodium vivax N -Myristoyltransferase Using Pyrazole-Derived Inhibitors.

  • Authors : Rodríguez-Hernández D; Department of Chemistry and Molecular Biology, University of Gothenburg, S-405 30 Gothenburg, Sweden.; Department of Structural and Functional Biology, Synthetic Biology Laboratory, Institute of Biology, University of Campinas, Campinas, SP 13083-862, Brazil.

Subjects: Pyrazoles*/Pyrazoles*/Pyrazoles*/chemistry ; Pyrazoles*/Pyrazoles*/Pyrazoles*/pharmacology ; Pyrazoles*/Pyrazoles*/Pyrazoles*/chemical synthesis

  • Source: Journal of medicinal chemistry [J Med Chem] 2024 May 09; Vol. 67 (9), pp. 7312-7329. Date of Electronic Publication: 2024 Apr 29.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

A Potential Multitarget Insect Growth Regulator Candidate: Design, Synthesis, and Biological Activity of Novel Acetamido Derivatives Containing Hexacyclic Pyrazole Carboxamides.

  • Authors : Guo B; Innovation Center of Pesticide Research, Department of Applied Chemistry, College of Science, China Agricultural University, Beijing 100193, China.; Chen L

Subjects: Insecticides*/Insecticides*/Insecticides*/chemistry ; Insecticides*/Insecticides*/Insecticides*/pharmacology ; Insecticides*/Insecticides*/Insecticides*/chemical synthesis

  • Source: Journal of agricultural and food chemistry [J Agric Food Chem] 2024 May 08; Vol. 72 (18), pp. 10271-10281. Date of Electronic Publication: 2024 Apr 24.Publisher: American Chemical Society Country of Publication: United States NLM ID: 0374755 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Design, synthesis and evaluation of a pyrazolo[3,4-d]pyrimidine derivative as a novel and potent TGFβ1R1 inhibitor.

  • Authors : Wang Y; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin, 300071, PR China.; Liu Y

Subjects: Receptor, Transforming Growth Factor-beta Type I*/Receptor, Transforming Growth Factor-beta Type I*/Receptor, Transforming Growth Factor-beta Type I*/antagonists & inhibitors ; Receptor, Transforming Growth Factor-beta Type I*/Receptor, Transforming Growth Factor-beta Type I*/Receptor, Transforming Growth Factor-beta Type I*/metabolism ; Drug Design*

  • Source: European journal of medicinal chemistry [Eur J Med Chem] 2024 May 05; Vol. 271, pp. 116395. Date of Electronic Publication: 2024 Apr 12.Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Safety and efficacy of zandelisib plus zanubrutinib in previously treated follicular and mantle cell lymphomas.

Subjects: Lymphoma, Mantle-Cell*/Lymphoma, Mantle-Cell*/Lymphoma, Mantle-Cell*/drug therapy ; Lymphoma, Follicular*/Lymphoma, Follicular*/Lymphoma, Follicular*/drug therapy ; Lymphoma, Follicular*/Lymphoma, Follicular*/Lymphoma, Follicular*/mortality

  • Source: British journal of haematology [Br J Haematol] 2024 May; Vol. 204 (5), pp. 1762-1770. Date of Electronic Publication: 2024 Mar 19.Publisher: Wiley-Blackwell Country of Publication: England NLM ID: 0372544 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

A pragmatic guide for management of adverse events associated with lorlatinib.

  • Authors : Liu G; Princess Margaret Cancer Centre, University Health Network, Toronto, ON, Canada. Electronic address: .; Mazieres J

Subjects: Lactams*/Lactams*/Lactams*/adverse effects ; Aminopyridines*/Aminopyridines*/Aminopyridines*/adverse effects ; Aminopyridines*/Aminopyridines*/Aminopyridines*/therapeutic use

  • Source: Lung cancer (Amsterdam, Netherlands) [Lung Cancer] 2024 May; Vol. 191, pp. 107535. Date of Electronic Publication: 2024 Mar 15.Publisher: Elsevier Scientific Publishers Country of Publication: Ireland NLM ID: 8800805 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Novel Pyrazole-4-Carboxamide Derivatives Containing Oxime Ether Group as Potential SDHIs to Control Rhizoctonia solani .

  • Authors : Luo B; College of Life Sciences, Xinyang Normal University, Tea Plant Biology Key Laboratory of Henan Province, Xinyang 464000, China.; Wu Y

Subjects: Rhizoctonia*/Rhizoctonia*/Rhizoctonia*/drug effects ; Rhizoctonia*/Rhizoctonia*/Rhizoctonia*/growth & development ; Fungicides, Industrial*/Fungicides, Industrial*/Fungicides, Industrial*/pharmacology Rhizoctonia solani; Sclerotinia sclerotiorum; Botrytis cinerea

  • Source: Journal of agricultural and food chemistry [J Agric Food Chem] 2024 May 01; Vol. 72 (17), pp. 9599-9610. Date of Electronic Publication: 2024 Apr 22.Publisher: American Chemical Society Country of Publication: United States NLM ID: 0374755 Publication Model: Print-Electronic Cited Medium: Internet

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  • 1-10 of  69,166 results for ""Pyrazoles""